Noj qab haus huv, Npaj
"Felodip": cov lus qhia rau kev siv, xyuas. tshuaj analogues
Uas hu rau cov tshuaj "Felodip"? Cov lus qhia rau kev siv ntawm cov tshuaj yuav tau piav nyob rau hauv kom meej nyob rau hauv lub hais tsab xov xwm. Tsis tas li ntawd tawm ntawm nws, koj yuav kawm txog dab tsi tshuaj no yog muab, dab tsi phiv nws muaj, seb puas los yog tsis cov tshuaj no contraindications, ntau npaum li cas nws cov nqi, uas muaj analogues thiab li ntawd.
Muaj pes tsawg leeg ntawm yeeb tshuaj, ib daim ntawv ntawm manufacturing thiab lub ntim
Nyob rau hauv dab tsi tau daim ntawv nyob rau ntawm lub tsev muag tshuaj tshuaj "Felodip"? nyob rau kev siv ntawm cov tshuaj no daim ntawv qhia hais tias nws yog muaj nyob rau hauv daim ntawv ntawm cov ntsiav tshuaj nrog heev kev txiav txim. Ntxiv mus, ntau koob tshuaj ntawm cov tshuaj muaj ib tug txawv lub hnab ntawv:
- daj tshuaj nyob rau hauv daim ntawv ntawm cov lentils, tsis muaj tsw denoted los ntawm tus xov tooj 2.5. Lub active caij xws tshuaj felodipine ua nyob rau hauv ib tug npaum li ntawm 2.5 mg. Cam ntawm cov tshuaj yog lactose monohydrate, hypromellose, microcrystalline cellulose, liab hlau oxide, povidone, titanium dioxide, propyl gallate, daj hlau oxide, magnesium stearate, propylene glycol, anhydrous colloidal silica, talc. Nyob rau hauv lub qhov muag ntawm active tshuaj nkag mus rau hauv sawv hlwv 10 ntsiav tshuaj uas yog muab tso rau hauv cov duab los qhia thawv.
- Ntsiav tshuaj ntawm lub teeb liab xim nyob rau hauv tus duab ntawm lentils, tsis muaj tsw denoted los ntawm tus xov tooj 5. Lub active tivthaiv xws npaj protrudes felodipine nyob rau hauv ib tug npaum li ntawm 5 mg. Cam ntawm cov tshuaj protrude lactose monohydrate, hypromellose, microcrystalline cellulose, liab hlau oxide, povidone, titanium dioxide, propyl gallate, daj hlau oxide, magnesium stearate, propylene glycol, anhydrous colloidal silica, talc. Nyob rau hauv lub qhov muag ntawm active tshuaj nkag mus rau hauv sawv hlwv 10 ntsiav tshuaj, yog muab tso rau hauv cov duab los qhia thawv.
- Ntsiav tshuaj liab xim av lentil zoo li tus tsis muaj tsw xaiv tus nab npawj 10. Lub active caij ntawm xws li ib tug yeeb tshuaj felodipine ua nyob rau hauv ib tug npaum li ntawm 10 mg. Koom Haum yog lactose monohydrate, hypromellose, microcrystalline cellulose, liab hlau oxide, povidone, titanium dioxide, propyl gallate, daj hlau oxide, magnesium stearate, propylene glycol, anhydrous colloidal silica, talc. Nyob rau hauv lub qhov muag ntawm active tshuaj nkag mus rau hauv sawv hlwv 10 ntsiav tshuaj. Hlwv muab tso rau hauv cov duab los qhia thawv.
Lub pharmacological thaj chaw ntawm cov tshuaj
Yuav ua li cas yog ib tug kho mob ntaus ntawv "Felodip"? Cov lus qhia rau kev siv ntawm cov tshuaj hais tias nws yog ib tug poov hlau channel blocker qeeb. Saib cov tshuaj belongs rau cov pab pawg neeg ntawm dihydropyridine.
Cov tshuaj no yog muaj peev xwm mus pheev antianginal thiab antihypertensive los. Nyob rau hauv tas li ntawd, nws thiaj li lub siab (cov ntshav) los ntawm zuj zus lawm peripheral vascular kuj.
Yuav ua li cas lwm yam khoom muaj tshuaj "Felodip"? Cov lus qhia rau kev siv ntawm cov kev npaj muaj cov ntaub ntawv hais tias nws muaj ib koob tshuaj-dependent anti-ischemic nyhuv. Tshuaj thiaj li infarction loj, me, thiab tseem tiv thaiv lub cev los ntawm reperfusion teeb meem.
Qhov cuab yeej no muaj suab tsis muaj tsis zoo inotropic nyhuv. Nws muaj ib tug tsawg heev nyob rau hauv kev system.
Cov tshuaj ntawm cov tshuaj
Yuav ua li cas ntev cov tshuaj yog absorbed, "Felodip"? Cov lus qhia rau kev siv, qhov no tswv yim txhais tau tias muab hais tias tom qab txhaj ib koob tshuaj medicament mus rau hauv lub active tshuaj yog yuav luag tag absorbed los ntawm cov hnyuv thiab ua sai li sai tau. Tsaug rau nws cov tshuaj daim ntawv no, ncua kev tso tawm ntawm lub active caij kom nws niaj hnub concentration hauv cov ntshav (nyob rau hauv ib hnub), thiab kuj ua rau yus mus rau ib qho kev nce rau hauv lub nqus theem.
Peb tsis tau hais tias cov bioavailability ntawm cov tshuaj tsis yog nyob ntawm seb kho koob thiab yog kwv yees li 15%.
Ruaj rau ntshav cov nqaijrog thiab ntau precisely nws yog kwv yees li 99%. Lub medicament yog tso tawm nrog rau mis mis nyuj thiab penetrates cov ntshav-hlwb barrier thiab cov placental barrier. Nrog heev siv cov active tshuaj tsis muaj txuam nrog no tshwm sim.
Qhov twg cov tshuaj yog metabolized "Felodip"? Lub active ingredient ntawm no neeg sawv cev yog metabolized nyob rau hauv lub siab. Nyob rau hauv daim ntawv no tsaug zog metabolites.
Lub ib nrab-lub neej ntawm cov tshuaj yog hais txog 25 teev. Tso tawm kom pom kev npaj raws li metabolites (kwv yees li 70%) nyob rau hauv cov zis thiab feces (30%).
indications medicament
Nyob rau hauv tej rooj plaub, tus neeg mob yog tshuaj "Felodip" (5 mg) Cov lus qhia ntawm cov tshuaj no muaj cov nram qab no daim ntawv teev cov indications rau kev siv:
- tawg;
- angina;
- arrhythmia;
- coronary mob plawv;
- lub plawv mob;
- Raynaud lub syndrome.
Contraindications tshuaj
Nyob rau hauv uas tus neeg mob yog nruj me ntsis txwv tsis pub noj tshuaj "Felodip"? Xyuas ntawm cov kws kho mob, raws li tau zoo raws li lub nrog cov lus qhia teev tias cov tshuaj yuav tsum tsis txhob yuav siv nyob rau hauv cov nram no tej yam kev mob:
- mob myocardial infarction, raws li zoo raws li nyob rau ib lub hlis tom qab myocardial;
- tsis ruaj tsis khov angina;
- cardiogenic poob siab;
- lub plawv tsis ua hauj lwm, tshwj xeeb tshaj yog decompensated;
- aortic stenosis (clinically tseem ceeb);
- cev xeeb tub;
- hypotension (mob loj heev);
- nyob rau hauv cov me nyuam thiab cov tub ntxhais hluas (nyob rau hauv 18 xyoo);
- thaum lub sij hawm lactation;
- nce rhiab heev ntawm tus neeg mob mus rau yeeb tshuaj los yog lwm yam dihydropyridine derivatives.
Ib tug yuav tsum tsis nco qab txog tias qhov cuab tam nrog huab ceev faj tshuaj rau cov neeg mob nrog hepatic thiab raum insufficiency.
Medical ntaus ntawv "Felodip": cov lus qhia rau kev siv
Analogues ntawm no lub cuab tam yuav tsum tau nthuav tawm ib me ntsis ntxiv. Tam sim no kuv xav qhia rau koj txog yuav ua li cas cov tshuaj yuav tsum tau coj kom raug.
Thaum tawg koob tshuaj rau cov neeg laus thiab cov neeg laus cov neeg yog teem ib lub zuj zus. Feem ntau, thawj zaug nqi ntawm cov tshuaj yog 5 mg ib zaug ib hnub twg. Thaum lub sij hawm xaiv uas tsim nyog cov neeg mob ntau npaum yog pom zoo kom siv cov ntsiav tshuaj ntawm 2.5 mg. Thaum lub ceev yuav tsum ua kom lub koob tshuaj yuav ua tau. Qhov nruab nrab lub ntim ntawm ib tug medicament rau tus txij nkawm kev kho mob ntawm 5-10 mg ib hnub twg.
Rau cov neeg laus cov neeg mob los yog cov neeg mob uas tsis hnov lub siab muaj nuj nqi nyob rau hauv thaum ntxov tshuaj kho yog muab nyob rau hauv ib tug npaum li ntawm 2.5 mg ib hnub twg.
Nyob rau hauv ruaj khov angina tshuaj "Felodip" tshuaj ib lub zuj zus. Yog li nws pib koob tshuaj (rau cov neeg laus) yog 5 mg ib zaug ib hnub twg. Yog hais tias yuav tsum tau, lub koob tshuaj yuav tau nce mus rau 10 mg ib hnub twg. Qhov siab tshaj plaws txhua txhua hnub ntau npaum li cas ntawm cov tshuaj yog 20 mg.
Ntsiav tshuaj "Felodip" yog tso cai rau coj nyob rau hauv ua ke nrog nrog ACE inhibitors, beta-blockers thiab diuretics. Txawm li cas los, nws yuav tsum tau muab sau tseg tias thaum lub hypotensive cov nyhuv yog kho kom zoo. Yog li ntawd koj yuav tsum tau ceev faj heev vim hais tias ntawm qhov raug mob ntawm hypotension.
Nyob rau hauv cov neeg mob uas muaj mob loj siab muaj nuj nqi rau hauv lub koob tshuaj yuav tsum raug txo.
Xa los ntawm cov tshuaj yuav tsum tsuas yog noj nyob rau hauv thaum sawv ntxov ua ntej noj tshais. Nyob rau hauv cov ntaub ntawv no, cov ntsiav tshuaj nyob rau hauv txhua rooj plaub nws yog tsis yooj yim sua kom keej, crush los yog sib faib.
overdose txhais tau tias
Tsis yog kev siv cov tshuaj "Felodip" li nram qab no cov tsos mob ntawm overdose yuav tshwm sim nyob rau hauv cov neeg mob: bradycardia thiab hypotension (mob loj heev).
Nyob rau hauv cov ntaub ntawv ntawm tshwm sim ntawm tej tsos mob symptomatic txoj kev kho. Yog hais tias hypotension (mob loj heev) cov neeg mob muab ib tug kab rov tav txoj hauj lwm thiab nqa ob txhais ceg. Nrog rau kev hwm mus bradycardia, nyob rau hauv uas cov ntaub ntawv rau tus neeg mob atropine intramuscularly xeem nyob rau ib ntau npaum ntawm 0.5-1 mg. Yog hais tias tsim nyog, kom tau qhov ntim ntawm ntshav Txoj kev lis ntshav yog nqa tawm nrog sodium chloride, piam thaj tov los yog dextran.
Thaum lub saum toj no-piav inefficiency ntsuas tshuaj rau ib tug neeg mob nrog ib tug predominant ntxim rau cov alpha-adrenergic receptors.
Sab los los ntawm kev noj cov tshuaj
Tau ib tug tsis zoo feem nyob rau tib neeg lub cev kev noj cov tshuaj "Felodip"? Analogues ntawm no lub cuab tam thiab kev npaj nws tus kheej feem ntau ua rau mob taub hau, lub ntsej muag yaug kais dej, kiv taub hau, palpitations thiab qaug zog. Txawm li cas los, nws yuav tsum tau muab sau tseg hais tias xws li kev tshua yog reversible. Lawv feem ntau yog tshwm sim nyob rau thaum pib ntawm txoj kev kho, raws li tau zoo raws li los ntawm nce lub tshuaj ntawm cov tshuaj.
Los ntawm txoj kev, nyob ntawm seb tus nqi tau txais tshuaj tus neeg mob tej zaum yuav tshwm sim thiab peripheral edema. Raws li kws txawj, lawv yog cov tshwm sim ntawm precapillary vasodilation.
Nyob rau hauv cov neeg mob uas ncig los yog pos hniav mob nyob rau hauv cov neeg mob uas tau txais cov tshuaj tej zaum yuav ua tau ib tug me me o ntawm cov pos hniav. Qhov no txoj kev muaj peev xwm yuav tiv thaiv tau, yog tias koj pom txhij txhua qhov ncauj.
Nyob rau hauv tej zaum peb yuav xav tias yuav tau txais cov tshuaj yuav ua kom muaj raws li nram no phiv:
- Plawv system: palpitations, tachycardia, thiab peripheral edema.
- Dermatological tshua: photosensitivity, pruritus, urticaria.
- Peripheral thiab central tshee system: paresthesia, mob taub hau thiab kiv taub hau.
- Licas: arthralgia, myalgia.
- Hnyuv: gingival hyperplasia, xeev siab, nce nyob rau hauv daim siab enzymes.
- Lwm yam: nkees, npau taws me ntsis kev tshua, xws li angioedema.
Analogs, thiab tus nqi ntawm cov tshuaj
Yuav ua li cas npaum li cas yog cov tshuaj ua ntej peb? Qhov ntawd yog qhov teeb meem tsa los ntawm ntau tus neeg mob niaj no kev kho mob raug muab. Nws yuav tsum tau muab sau tseg tias hnub no yog ib yam tshuaj yuav tau muas ntawm qhov nqi:
- Ntsiav tshuaj ntawm 2.5 mg (30 pieces) - 425 Lavxias teb sab rubles;
- ntsiav tshuaj nyob rau hauv ib tug ntim ntawm 5 mg (30 pieces) - 556 Lavxias teb sab rubles;
- ntsiav tshuaj nyob rau hauv ib tug ntim ntawm 10 mg (30 pieces) - 831 Lavxias teb sab rubles.
Yuav ua li cas yuav hloov tau cov tshuaj "Felodip"? Analogs ntawm cov tshuaj no yog muaj nyob rau hauv txhua lub chaw muag tshuaj. Ntawm lawv, kuv xav mus rau ntsiab li nram qab no tshuaj: "Plendil," "Felodipine-NW", "Felodipine" thiab "Felotenz retard."
Zoo tswv yim los ntawm cov neeg mob txog lam khoom
Testimonials txog "Felodip" npaj lub xeev hais tias nws yog zoo heev thiab zoo-taus los ntawm cov neeg mob, tsis hais hnub nyoog thiab yog txivneej los pojniam. Tsis tas li ntawd, active tshuaj tej zaum yuav tsum tau noj twb yog los ntawm cov neeg mob uas mob ntshav qab zib, raum mob, mob hawb pob thiab lwm yam obstructive ntsws kab mob nrog Raynaud lub syndrome, hyperlipidemia, gout, thiab tom qab mob ntsws hloov.
Muaj ntau cov kws txawj taw tes kom paub qhov tseeb hais tias cov tshuaj muaj tsis ntxim rau cov lipid profile thiab cov ntshav piam thaj concentration.
tsis zoo xyuas
Ntawm cov tsis zoo xyuas uas tawm cov neeg mob nyob rau hauv cov tshuaj no, peb yuav nco ntsoov cov neeg muaj feem xyuam rau cov nqi ntawm cov tshuaj. Txawm tias pharmacists cam hais tias nws tus nqi yog tag nrho raws li efficiency thiab zoo.
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