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"Brilint": kev piav qhia txog cov tshuaj, cov kev qhia ntawv. Analog "Brilinta"

"Brilint" - ib tug yeeb tshuaj uas yog dav siv nyob rau hauv kev phais thiab Cardiology, raws li muaj ankoagulyantnym thiab antiplatelet los. Nyob rau hauv feem ntau tus neeg mob, siv tau rau lub hom phiaj cupping angina (tsis ruaj tsis khov daim ntawv no) thiab ischemic mob, raws li tau zoo raws li ib tug prophylactic tus neeg saib xyuas tiv thaiv los ntshav tam sim ntawd ua ntej phais.

Qauv thiab pes tsawg leeg

Qhov "Brilinta" 90 mg (kuj analog) ntsiav tshuaj. Lawv yuav them rau ib zaj duab xis cover ntawm ib tug yellowish Hawj txawm. Zoo round biconvex.

Lub ntsiab active ingredient ntawm cov tshuaj yog ticagrelor. Cov adjuvants emit:

  • mannitol;
  • magnesium stearate;
  • calcium hydrogenphosphate;
  • sodium carboxymethyl cov hmoov txhuv nplej;
  • giproloza.

Tus zaj duab xis, nyob rau hauv lem, muaj hypromellose, talc, titanium dioxide, macrogol, zas xim (daj oxide).

Lub ntsiab nyhuv ntawm cov tshuaj

"Brilint" muaj antiplatelet txiav txim, i.e. tiv thaiv aggregation ntawm cov ntshav txhaws. Raws li ib tug tshwm sim ntawm lub ntsiab active tshuaj tivthaiv - ticagrelor - platelets poob lub peev xwm los lo ua ke, thiab yog li tsim txhaws.

Heev heev cov kev tshawb fawb paub meej tias qhov tseeb hais tias cov qauv ntawm cov "Brilinta" zoo tshaj nyob rau hauv ua ke nrog nrog salicylic acid. Analogichinye pom zoo thiab hais txog analogue "Brilinta" - "Plavix". Nyob rau hauv cov kev nyuaj siab muab kev koom tes cov neeg mob uas tus kab mob plawv nyob rau hauv hnub nyoog sib txawv pab pawg, thiab coj tus account ntawm lawv cov luj, txiv neej pw.

Lub hom phiaj ntawm txoj kev kho siv hais tias cov khoom - txo txoj kev pheej hmoo ntawm kev tuag, uas tej zaum yuav tshwm sim los ntawm ib tug malfunction ntawm cov hlab plawv system, tshwj xeeb yog angina pectoris thiab myocardial infarction.

indications

Txais tos "Brilinta" yog muaj nyob rau hauv cov ntaub ntawv ntawm qhov yuav tsum tau rau kom cov ntshav txhaws, xws li cov kev tiv thaiv ntawm cov teeb meem ntawm cov hlab plawv tus kab mob nyob rau hauv daim ntawv ntawm cov thrombosis thiab thromboembolism. Uas yog vim li cas cov tshuaj no yog qhia rau:

  • tsis ruaj tsis khov angina (Qhov no pathology yog yus muaj los ntawm deterioration ntawm cov ntshav ncig mus rau lub plawv mob, uas hawv ua phem myocardial);
  • myocardial infarction (tuag ntawm ib feem ntawm lub plawv);
  • kev ua tau zoo phais haujlwm rau lub coronary hlab ntsha ntawm lub plawv mob (thaum lub sij hawm percutaneous coronary tiv thaiv, los yog coronary artery bypass phais).

Nyob rau hauv tas li ntawd mus ncaj pov thawj, mus rau "Brilint" kev txiav txim ntawm tus kws kho mob tej zaum yuav tau tsa nyob rau hauv thiaj li yuav txo thrombosis nyob rau hauv lwm yam pathological tej yam kev mob, xws li thaum dissemirovannom intravascular coagulation.

Contraindications

Muaj ib tug xov tooj ntawm cov kev txwv, nyob rau hauv uas ntawm kev siv ntawm "Brilinta" yog tsis tau tso cai. Cov muaj xws li:

  • idiosyncrasy, xws li npau taws me ntsis rau lub active tshuaj los yog yam tsawg ib tug ntxiv koponentu;
  • active los ntshav, kev coj tus kheej pathological;
  • haemorrhagic stroke duab uas tau tsiv ua ntej lawm;
  • txo hepatocyte kev ua si, tiv thaiv uas muaj lub siab tsis ua hauj lwm;
  • koom haum saib xyuas ntawm cov tshuaj, lub ntsiab kev txiav txim ntawm uas muaj nyob rau hauv inhibition ntawm cov enzyme CYP3A4 ( «clotrimazole," "Ritonavir", "nefazodone");
  • Cov me nyuam mus txog hnub nyoog 18 xyoo;
  • thaum lub sij hawm cev xeeb tub thiab lactation.

Nyob rau hauv lub qhaj ntawv ntawm contraindications yuav tsum ua ua ntej pib ntawm txoj kev kho nrog cov tshuaj no.

Cov lus qhia rau kev siv

Muab "Brilint" yuav tsum nyob rau hauv lub tag nrho, cov tshuaj yuav tsum tsis txhob yuav chewed. Siv cov tshuaj tsis yog nyob ntawm seb lub sij hawm ntawm haus. Ntsiav tshuaj yuav tau haus ib tug me me npaum li cas ntawm cov kua.

Pom zoo ntau npaum: 1 ntsiav tshuaj ib hnub twg. Nws yog ib qho tseem ceeb noj cov tshuaj txhua txhua hnub nyob rau tib lub sij hawm.

Hoob no ntawm txoj kev kho nrog rau cov kev siv ntawm "Brilinta" (hloov yuav ua ntev) koj yuav tsum tau pib nrog ib tug muab ob npaug rau koob tshuaj (ob ntsiav tshuaj nyob rau hauv thawj hnub), thiab ces txav mus rau ib tug ib koob tshuaj ntawm 90 mg. Nyob rau hauv cov ntaub ntawv ntawm lub nkag ntawm cov tshuaj yuav tsum tsis txhob siv ib tug muab ob npaug rau koob tshuaj. Hnub tom qab ntawd tom qab ib tug tsis rov pib dua qub txais tos "Brilinta." Txawm li cas los, tej lub sijhawm yuav tsum tau zam.

Qhov nruab nrab ntev ntawm kev kho mob - 12 lub hlis.

Nyob rau hauv tas li ntawd, cov pom zoo simultaneous acetylsalicylic acid.

phiv

Ntawm cov atypical ces tau txais distinguished:

  • muaj zog heev yuav txo tau ntawm cov ntshav txhaws nrog txoj kev loj hlob ntawm kev txawv txav los ntshav;
  • kev tsis haum tshuaj;
  • xeev siab;
  • ntuav.

Thaum tshwm sim los ntawm cov tshuaj yuav tsum tau nres sai li sai tau.

overdose

Nyob rau hauv cov ntaub ntawv ntawm cov hauv qab no cov tsos mob tej zaum yuav tshwm sim tau txais ntau zog koob tshuaj ntawm cov tshuaj:

  • xeev siab;
  • tsam plab;
  • los ntshav;
  • kev cuam tshuam ntawm lub plawv.

Thaum lawv tshwm sim koj yuav tsum tsis txhob noj cov tshuaj, los pais plab lavage, hnyuv, thiab symptomatic txoj kev kho.

analogs

Thaum impossibility ntawm kev cov tshuaj yuav tsum tau paub dab tsi los hloov "Brilintu". Ntawm cov ntsiab counterparts sawv tawm:

  1. "Zilt". Qhov no analogue "Brilinta" nqi sib txawv, tab sis cov teebmeem ntawm ob tshuaj zoo sib xws thiab tswj cov kev tiv thaiv ntawm thrombosis. Active muaj yog clopidogrel. Lub indications rau cov kev siv ntawm cov nyiaj yog myocardial infarction, coronary syndrome, mob stroke, atrial fibrillation, coronary artery kab mob okklyuizonnaya. "Zilt" yog yus muaj los ntawm ib tug tsawg sab nyhuv.
  2. "Plavix". "Brilinta" los yog "Plavix" - uas yog ib qho zoo? Hais mas nws yeej tsis. Cov tshuaj yog txawv active tshuaj, tab sis cov nyhuv lawv muaj zoo sib xws. Qhov no pub rau siv ceev xwmphem lub chav kawm ntawm kev kho yog lwm txhais tau tias mus ntxiv kev kho mob nrog lwm tus. Analogue "Brilinta" "Plavix" yog muab rau cov neeg mob uas muaj atherosclerotic phenomena pom tias, cov neeg mob tom qab koj lub plawv nres thiab hlab ntsha tawg. Qhov no tshuaj yog tseem pheej yig dua analog. Yuav ua li cas mus xaiv: "Brilinta" los yog "Plavix". Uas yog zoo dua? Qhia ib tug kws kho mob.
  3. "Lopirel". Qhov no analogue "Brilinta" ua rau lub hauv paus ntawm clopidogrel, uas yog vim li cas qhov kev txiav txim yog raws kev coj kom platelets, tiv thaiv lawv lo ua ke. Tsis zoo li lwm txoj kev, "Lopirel" tej zaum yuav cuam tshuam rau functionality ntawm lub paj hlwb, ua pa licas, raws li zoo raws li ntawm hematopoiesis. Nyob rau hauv tas li ntawd, nws yog ib nqi nco ntsoov hais tias qhov no analogue tshuaj "Brilinta" yog tsis thawj, thiab cov generic, uas yog ib daim qauv ntawm "Plavix".

Nyob rau hauv tas li ntawd mus rau cov analogues tso cai rau kev siv ntawm lwm yam tshuaj uas muaj xws li cov teebmeem, tab sis txawv hom ntawm kev txiav txim ( "Cardiomagnyl", "Aspekard", "Tshuaj aspirin cardio").

Cov ntsiab lus uas thiab tej yam kev mob ntawm cia

Txee lub neej "Brilinta" (cov lus hais txog nws yuav luag tag nrho cov zoo) yog 2 xyoo. Yog li ntawd nws yog tsim nyog los soj ntsuam cov kub tsoom fwv (lub chav tsev nyob qhov twg lub muab neeg sawv cev yuav tsum muaj tsawg tshaj li 30 degrees, yuav tsum muaj tsis muaj lub teeb thiab dej). Nyob rau hauv tas li ntawd, lub cuab tam yuav tsum tau muaj kev tiv thaiv los ntawm cov me nyuam.

Nco ntsoov hais tias tag nrho cov kev teem caij yuav tsum ua kws kho mob.

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