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Angiotensin receptor blockers 2: tshuaj thiab mechanisms kev txiav txim ntawm

Ob kev tiv thaiv thiab kev kho mob ntawm cov hlab plawv tus kab mob yuav tsum tau ib tug luag hauj lwm thiab loj mus kom ze. Tej teeb meem yog nce kev txhawj xeeb txog cov neeg niaj hnub no. Yog li ntawd, muaj coob tus neeg yuav los kho lawv ntau maj mam. Xws li tus neeg muaj feem ntau yog kiag li las mees qhov yuav tsum tau mus yauv mus kho mob los yog noj tshuaj tsis muaj ib tug kws kho mob tshuaj (nyob rau lub tswv yim ntawm cov phooj ywg). Txawm li cas los, nws yog ib qho tseem ceeb rau koj nco ntsoov tias ib txhia tshuaj pab lwm tus neeg, nws tsis lav hais tias nws yuav pab tau koj. Rau lub tsim ntawm kev kho mob kiag yuav tsum tau txaus paub, kev txawj ntse, uas tsuas muaj cov kws tshwj xeeb. Tsis tas li ntawd muab tej tshuaj yuav tsuas xaiv cov neeg tus yam ntxwv ntawm tus neeg mob, tus heev ntawm tus kab mob no, tshwj xeeb tshaj yog thaum kawg nws thiab keeb kwm. Ntxiv mus, niaj hnub no muaj ntau ntau yam zoo tshuaj uas raug xaiv thiab raug tsa los tsuas cov tub txawg ua tau. Piv txwv li, nws yog hais txog sartans - tshwj xeeb cov pab pawg neeg ntawm cov tshuaj (kuj hu ua angiotensin receptor blockers 2). Yuav ua li cas yog cov tshuaj? Yuav ua li cas ua lub angiotensin receptor 2? Contraindications rau kev siv ntawm tshuaj mus rau uas pawg paitsentov? Nyob rau hauv tej rooj plaub, nws yuav tsim nyog rau siv lawv? Uas tshuaj muaj nyob rau hauv pab pawg neeg no tej? Cov lus teb rau cov no thiab lwm cov lus nug yuav tsum los sib tham nyob rau hauv no tsab xov xwm.

Sartana

Xam tias yog raws li ib pab pawg neeg ntawm tshuaj yog muaj npe raws li nram no: angiotensin receptor blockers 2. Formulations ntawm no pab pawg neeg ntawm cov tshuaj, peb tau ua los ntawm ceev faj txoj kev tshawb no ntawm cov ua ntawm cov kab mob ntawm cov hlab plawv system. Niaj hnub no, lawv siv nyob rau hauv Cardiology yog ua ntau heev.

Angiotensin receptor 2: mechanisms ntawm kev txiav txim

Ua ntej koj yuav pib siv tshuaj, nws yog ib qho tseem ceeb kom nkag siab txog raws nraim yuav ua li cas lawv ua hauj lwm. Yuav ua li cas cuam tshuam rau tib neeg lub cev angiotensin receptor 2? Npaj ntawm no pab pawg neeg khi rau receptors, li no thaiv cov hlab ib tug tseem ceeb nce nyob rau hauv cov ntshav siab. Qhov no yuav pab tiv thaiv kom txhob zoo tawg. angiotensin receptor blockers 2 yog qhov zoo tshaj nyob rau hauv no hwm tshuaj. Kws txawj yog them vim cov xim rau lawv.

Classification: angiotensin receptor blockers 2

Muaj ob peb hom sartans uas txawv nyob rau hauv lawv cov tshuaj qauv. Nws yuav tau mus xaiv lub uas tsim nyog tus neeg mob angiotensin receptor blockers 2. yeeb siv tshuaj, uas yuav tsum tau teev tseg hauv qab no, nws yog ib qho tseem ceeb los mus tshawb nrhiav thiab sib tham txog qhov kev tsimnyog ntawm lawv cov kev siv nrog koj tus kws kho mob.

Yog li ntawd, muaj plaub pawg sartans:

  • Biphenyl tetrazole derivatives.
  • Nebifenilovye tetrazole derivatives.
  • Nebifenilovy netetrazol.
  • Tsis-cyclic tebchaw.

Yog li, muaj ntau ntau hom ntaub ntawv, uas yog cais los ntawm angiotensin 2. Formulations (tub ntxhais daim ntawv teev) receptors uas hais hauv qab no:

  • "Losartan".
  • "Eprosartan".
  • "Irbesartan".
  • "Telmisartan".
  • "Valsartan".
  • "Candesartan".

indications

Siv no pab pawg neeg ntawm tshuaj yuav tsuas yuav muab los ntawm ib tug kws kho mob. Muaj ntau ntau tus neeg mob nyob rau hauv uas nws yuav tsum tau tsim nyog mus siv angiotensin receptor blockers 2. Soj ntsuam yam ntawm no pab pawg neeg hauv qab no npaj:

  • Tawg. Hais tias yog, tus kab mob no yog ib tug loj yeej rau kev siv sartans. Qhov no yog vim lub fact tias angiotensin receptor blockers 2 tsis adversely cuam tshuam lub metabolism thiab tsis ua rau erectile kawg, bronchial tsis tsis tau permeability. Nyhuv ntawm cov tshuaj yuav pib tom qab ob mus rau plaub lub lis piam tom qab pib ntawm kev kho mob.
  • Lub plawv tsis ua hauj lwm. Angiotensin receptor blockers 2 inhibit qhov kev txiav txim ntawm lub renin-angiotensin-aldosterone system, uas nws ua si thiab provokes tus txoj kev loj hlob ntawm tus kab mob.
  • Nephropathy. Vim mob ntshav qab zib mellitus thiab tawg, muaj yeej loj heev teeb nyob rau hauv lub hauj lwm ntawm ob lub raum. angiotensin receptor blockers 2 tiv thaiv cov hauv nruab nrog cev thiab yog tsis muaj peev xwm mus tso saib ntau heev protein nyob rau hauv cov zis.

"Losartan"

Pib tshuaj muaj nyob rau hauv cov pab pawg neeg ntawm sartans. "Losartan" - blocker, angiotensin-2 receptor Nws txim hluav taws xob los ntawm lwm yam tshuaj yog ib tug tseem ceeb nce nyob rau hauv ce kam nyob rau hauv tib neeg kev txom nyem los ntawm lub plawv tsis ua hauj lwm. Los ntawm cov tshuaj yuav lub siab tshaj plaws twb tom qab rau lub sij hawm ntawm kev noj cov tshuaj. Cov nyhuv yog mus txog tom qab peb los yog rau lub lim tiam ntawm cov tshuaj daim ntawv thov.

Lub ntsiab indications rau kev siv ntawm cov tshuaj nyob rau hauv kev saib xyuas no muaj raws li nram no:

  • lub plawv tsis ua hauj lwm;
  • tawg;
  • yuav txo tau nyob rau hauv txoj kev pheej hmoo ntawm stroke nyob rau hauv cov neeg mob uas muaj cov prerequisites rau qhov no.

Koj yuav siv tsis tau "Losartan" thaum lub sij hawm nyuam thiab thaum lub sij hawm pub niam mis, raws li zoo raws li nyob rau hauv cov ntaub ntawv ntawm ib tug neeg kev mloog tau tus neeg lub Cheebtsam ntawm cov kev npaj.

angiotensin receptor blockers 2, uas siv rau qhov suav hais tias cov tshuaj yuav ua rau ib txhia phiv xws li kiv taub hau, insomnia, pw tsaug zog ua cuam tshuam, saj, tsis pom kev, co, kev nyuaj siab, nco tsis meej, pharyngitis, hnoos, bronchitis, rhinitis, xeev siab, gastritis, mob hniav, raws plab, anorexia, ntuav, tu-sauv, mob caj dab, mob nyob rau hauv lub xub pwg, rov qab, ob txhais ceg, palpitations, anemia, lub raum tsis ua hauj lwm, impotence, weakening ntawm libido, erythema, alopecia, tawm pob, khaus, o, ua npaws, gout, hyperkalaemia .

Yuav tsum muab cov tshuaj ib hnub ib zaug, tsis hais pluas mov, lub koob tshuaj tshuaj los ntawm cov kws kho mob.

"Valsartan"

Tam sim no medicament yog zoo nyob rau hauv txo mob hypertrophy, uas tshwm sim vim txoj kev loj hlob ntawm tawg. Ntsoos ntsoos tsis tshwm sim tom qab discontinuation ntawm cov tshuaj, txawm hais tias nws muaj peev xwm ua rau ib txhia angiotensin receptor 2 (piav qhia sartans pab pawg neeg yuav pab tau nrhiav tau tawm raws nraim li cas mus tshuaj muaj xws li no feature).

Lub ntsiab indications rau tau txais cov tshuaj yeeb dej caw nyob rau hauv lo lus nug yog cov nram qab no tej yam kev mob: myocardial infarction, thawj los sis theem nrab tawg, txhaws lub plawv tsis ua hauj lwm.

Cov ntsiav tshuaj yog npaum li cas hais lus. Lawv yuav tsum tau nqos tsis zom. Koob appoints tus kws kho mob. Txawm li cas los, lub siab tshaj plaws nqi ntawm ib yam khoom uas yuav tsum tau noj thaum lub sij hawm hnub, yog rau puas thiab plaub caug milligrams.

Tej zaum nws yuav muaj nyob rau hauv lub cev thiab tus tsis zoo feem ntawm angiotensin receptor blockers 2. Sab teebmeem, uas yuav ua rau "Valsartan": tsis libido, khaus, kiv taub hau, neutropenia, tsis nco qab, sinusitis, insomnia, myalgia, raws plab, anemia, hnoos, mob nyob rau hauv lub rov qab , kiv tauv hau, xeev siab, vasculitis, edema, txhaws ntswg. Yog hais tias koj muaj tej yam ntawm cov tshuaj, koj yuav tsum tam sim ntawd sab laj ib tug tshwj xeeb.

"Candesartan"

Saib formulation formulated raws li cov ntsiav tshuaj rau qhov ncauj thawj coj. Nws yuav tsum tau coj ib zaug los yog ob zaug ib hnub twg nyob rau hauv tib tus nqi ntawm lub sij hawm tsis hais tus noj mov. Koj yuav tsum ua tib zoo ua raws li cov tswv yim pom zoo ntawm cov kws txawj. Nws yog ib qho tseem ceeb tsis txhob tsum tsis noj cov tshuaj, txawm tias koj xav tias zoo dua. Txwv tsis pub, nws yuav neutralize cov hauj lwm zoo ntawm cov tshuaj.

Thaum uas siv cov nws yuav tsum tau ceev faj rau cov neeg mob uas raug kev txom nyem los ntawm cov ntshav qab zib, raum insufficiency los yog daug lawm tus me nyuam. Tag nrho cov tej yam kev mob yuav tsum tau txais kev ceeb toom cov tub txawg.

"Telmisartan"

Xam tias yog ib tug yeeb tshuaj yog absorbed los ntawm tus mob huam nyob rau hauv ib tug ncaj luv luv lub sij hawm ntawm lub sij hawm. Nws yuav tsum noj tsis hais noj mov. Lub ntsiab hais txog kev siv yog tawg. Lub ib nrab-lub neej ntawm cov tshuaj yog ntau tshaj nees nkaum lub sij hawm. Lub tshuaj no yog muab tau los ntawm cov hnyuv yuav luag unchanged.

Txwv tsis pub muaj kev xeem ua xam tau tias yog tshuaj thaum lub sij hawm cev xeeb tub los yog pub niam mis.

Cov tshuaj yuav ua rau cov nram qab no tshwm sim tsis zoo: insomnia, kiv taub hau, xeev siab, diareyayu, kev nyuaj siab, mob plab, pharyngitis, tawm pob, hnoos, myalgia, mob txeeb zig, tsis tshua muaj ntshav siab, mob hauv siab, palpitations, anemia.

"Eprosartan"

Xam tias yog ib tug yeeb tshuaj yuav tsum tau noj ib zaug ib hnub twg. Cov pom zoo nqi ntawm cov tshuaj rau ib tug tib daim ntawv thov yog rau pua milligrams. Qhov siab tshaj plaws cov nyhuv yog tiav tom qab ob peb lub lis piam ntawm kev siv. "Eprosartan" yuav ua tau ib feem ntawm ib tug kev kho thiab monotherapy ntsiab tivthaiv.

Nyob rau hauv tsis muaj cov ntaub ntawv yuav tsis muab suav hais tias thov cov tshuaj thaum lub sij hawm lactation los yog cev xeeb tub.

Yuav ua li cas tshwm sim muaj tshwm sim thaum uas siv cov "eprosartan"? Ntawm lawv yog cov hauv qab no: tsis muaj zog, raws plab, kiv taub hau, mob taub hau, txhaws ntswg, hnoos, txog siav, edema, mob hauv siab.

"Irbesartan"

Saib cov tshuaj noj ntawm ncauj. Nws nyob hauv ib tug luv luv lub sij hawm yog absorbed los ntawm cov hnyuv ib ntsuj av. Qhov siab tshaj plaws concentration ntawm ib yam khoom nyob rau hauv cov ntshav no tshwm sim tom qab xwb ib tug ob peb teev. Khoom noj khoom haus kom tsawg tsis cuam tshuam rau miv nyuas siv zug ntawm cov tshuaj.

Yog hais tias tus neeg mob yog muab hemodialysis, nws tsis cuam tshuam rau mechanism ntawm qhov kev txiav txim "Irbesartan". Qhov no cov ntaub ntawv uas yog tsis muab los ntawm tib neeg lub cev los ntawm hemodialysis. Ib yam li ntawd, cov tshuaj yuav xyuam xim txais cov neeg mob kev txom nyem los ntawm mob npuas paug ntawm me me los yog muaj mob loj tsawv heev.

Cov tshuaj yuav tsum tau nqos tsis zom. Nws daim ntawv thov tsis yuav tsum tau ua ke nrog rau cov pluas noj. Pom starting koob yog suav tias yog ib puas thiab tsib caug milligrams ib hnub twg. Laus cov neeg mob kom pib kho mob nrog xya caum milligrams. Thaum lub sij hawm kev kho mob, koj tus kws kho mob tej zaum yuav txiav txim siab mus hloov ntau npaum (xws li, nws nce nyob rau hauv lub mob ntawm txaus los khi kho teebmeem nyob rau hauv lub cev). Nyob rau hauv cov ntaub ntawv no, tus neeg mob yuav tsum tau coj peb puas milligrams ntawm cov tshuaj los yog hloov cov thawj cov tshuaj nyob rau hauv tus. Piv txwv li, rau cov kev kho mob ntawm cov ntshav qab zib mellitus ntawm ob hom thiab tawg ntau npaum yuav tsum tau maj mam hloov los ntawm ib puas thiab tsib caug milligrams ib hnub twg rau peb puas milligrams (uas yog tus naj npawb ntawm medicament yog qhov zoo tshaj rau kev tswj nephropathy).

Muaj ntau yam nta ntawm daim ntawv thov ntawm cov tshuaj no. Yog li, cov neeg mob kev txom nyem los ntawm mob ntawm dej thiab mob electrolyte tshuav nyiaj li cas, ua ntej kev kho mob ntawm ib co ntawm nws cov ces yog tsim nyog los tshem tawm (hyponatremia).

Yog hais tias muaj yog ib tug ua txhaum ntawm lub raum muaj nuj nqi, nws kho mob regimen nyob rau hauv tib neeg tej zaum yuav tau tib yam li hais tias muaj yog tsis muaj xws teeb meem. Tib yam siv rau hepatic kawg me ntsis rau ntsis. Nyob rau tib lub sij hawm, thaum hemodialysis thawj zaug nqi ntawm cov tshuaj yuav tsum tau txo los ntawm ib nrab piv nrog rau cov pa thiab roos xya caum-tsib milligrams ib hnub twg.

Kws txawj tsis pom zoo kom siv ntawm qhov suav hais tias cov tshuaj rau cov menyuam yaus, vim nws tsis yog tsim raws li nws muaj kev ruaj ntseg thiab zoo nyob rau hauv no muaj hnub nyoog ntawm cov neeg mob.

"Irbesartan" nruj me ntsis contraindicated rau cov kev siv los ntawm cov poj niam uas tuav ib tug me nyuam, vim nws ncaj qha muaj feem xyuam rau tus txheej txheem ntawm me nyuam hauv plab kev loj hlob. Yog hais tias lub cev xeeb tub thaum lub sij hawm ntawm lawv cov kev kho, cov xeem yuav tsum raug rho tawm tam sim ntawd. Nws yog pom zoo kom hloov mus rau lwm txoj khoom ua ntej pib ntawm cev xeeb tub npaj. Saib txwv tsis pub siv yeeb tshuaj thaum lub sij hawm kev pub niam mis, raws li muaj yog tsis muaj ntaub ntawv raws li seb tus tshuaj nyob rau hauv niam cov kua mis.

Summing li

Kom koj noj qab haus huv - tus kheej luag hauj lwm ntawm txhua tus tib neeg. Thiab cov laus lub hnub nyoog, lub ntau kev rau siab nws yuav tau ua. Txawm li cas los, kev lag luam kws muaj lub invaluable pab, lossi ua hauj lwm los tsim ib tug zoo dua thiab zoo tshaj cov tshuaj. Xws li lug siv nyob rau hauv sib ntaus tawm tsam tus kab mob plawv thiab suav hais tias nyob rau hauv no tsab xov xwm, angiotensin receptor blockers 2. yeeb siv tshuaj, ib daim ntawv teev cov neeg uas tau raug nplua thiab sib tham nyob rau hauv kom meej nyob rau hauv no tsab xov xwm, yuav tsum tau siv thiab thov kom lo lus uas peb lub mus kawm tus kws kho mob uas yog zoo muaj cuab kav nrog tam sim no tus neeg mob lub xeev kev kho mob, thiab tsuas yog nyob rau hauv nws tas mus li tswj. Cov xws tshuaj yog cais "Losartan" "Eprosartan" "irbesartan" "telmisartan" "Valsartan" thiab "Candesartan". Muab tshuaj xam tau tias yog xwb nyob rau hauv cov nram no mob: nyob rau hauv lub xub ntiag ntawm tawg, mob raum tus kab mob thiab lub plawv tsis ua hauj lwm.

Yog hais tias qhov kev kawm, pib self-ib qho tseem ceeb yuav tsum paub txog cov kev txaus ntshai uas yog txuam nrog nws. Firstly, thaum uas siv cov tshuaj xam tau tias yog ib qho tseem ceeb kom meej soj ntsuam cov tshuaj thiab lub caij nws tom nyob rau qhov tam sim no mob ntawm tus neeg mob. Mus nqa tawm tag nrho cov txheej txheem no tsuas yog ib tug kws muaj peev xwm kom zoo. Txij li thaum tsuas muaj ib tug kws kho mob ua tau raws li kev soj ntsuam thiab cov kev tshwm sim ntawm analyses muab tsim nyog ntau npaum thiab kev kho mob regimen meej tsim. Tom qab txoj kev kho yog yuav tsum tau zoo xwb nyob rau hauv cov kev tshwm sim hais tias ib tug neeg mob yuav ua raws li tus kws kho mob pom zoo.

Nyob rau lwm cov tes, nws yog ib qho tseem ceeb nyob rau hauv txhua txoj kev pab rau kev txhim kho lawv tus kheej lub cev mob los ntawm raws li cov kev cai ntawm ib tug noj qab nyob zoo txoj kev ua neej. Cov neeg mob yuav tsum tau kom kho pw tsaug zog thiab wakefulness, kom muaj cov dej tshuav nyiaj li cas, thiab kho noj zaub mov zoo (tom qab tag nrho, tsis txaus cov zaub mov, tsis txhob muab lub cev nrog rau txaus tseem ceeb as-ham, yuav tsis tau rov qab nyob rau hauv ib tug ib txwm atherosclerosis).

Xaiv high-zoo tshuaj. Saib xyuas ntawm koj tus kheej thiab koj tus hlub. Nyob twj ywm noj qab nyob zoo!

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