Noj qab haus huv, Npaj
"Luminal": cov lus qhia rau kev siv ntawm cov me nyuam mos
Yuav ua li cas yog cov tshuaj "Luminal"? Cov lus qhia thiab indications ntawm cov tshuaj no yuav tsum tau tham hauv qab no. Peb kuj piav txog cov pharmacological thaj chaw ntawm cov tshuaj, nws tshwm sim thiab contraindications.
Muaj pes tsawg leeg ntawm cov tshuaj thiab hauv daim ntawv ntawm
Uas muaj ib tug yeeb tshuaj "Luminal"? Cov lus qhia rau kev siv qhia tias nyob rau hauv nyob tus yeees ntawm no formulation muaj xws li cov active ingredient xws li phenobarbital. Tsis tas li ntawd xam tau tias yog txhais tau tias muaj xws li cov nram qab no ntxiv Cheebtsam: qos starch, gelatin, talc thiab calcium stearate.
Kev npaj "Luminal", indications uas yog hais hereinafter, yog marketed nyob rau hauv daim ntawv ntawm ib tug hmoov npaj rau tov rau kev txhaj tshuaj. Tsis tas li ntawd qhov cuab tam yuav yuav nyob rau hauv daim ntawv ntawm cov ntsiav tshuaj ntawm 100 mg, uas yog tau ntim rau hauv lub cell contour thiab ntim ua los ntawm daim ntawv, ntsig txog.
Tus kho nyhuv ntawm cov tshuaj
Yuav ua li cas yog cov tshuaj raws li "Luminal"? Cov lus qhia rau kev siv cav hais tias qhov no tshuaj muaj sedative, hypnotic thiab anticonvulsant los.
Saib medicament muaj peev xwm ntawm exerting suppressive txiav txim (non-xim) nyob rau hauv tus tib neeg lub paj hlwb, thiab kuj inhibit tej cheeb tsam (feem ntau yog piav thoob hlo) cortex txo locomotor kev ua si, tsim nkees nkees thiab ua kom loog.
Tshuaj "Luminal" qhia ntawv nyob rau daim ntawv thov ntawm cov uas yog nyob rau hauv daim ntawv teeb yog ib tug heev haib barbiturate. Nws sedative-hypnotic zog yog vim inhibition ntawm cov kev ua ntawm lub hlwb, uas qhib lub reticular tsim ntawm lub nuclei ntawm lub thalamus, brainstem, li no inhibit sis ntawm hais tias lug nrog lub cerebral cortex.
nta tshuaj
Yuav ua li cas yog zoo tshaj plaws tshuaj "Luminal"? Cov lus qhia rau kev siv (cov me nyuam mos yog ib tug txhais tau tias tus kws kho ntau heev) hais tias pw tsaug zog los ntawm qhov no barbiturate, muab piv nrog saline muaj ib tug txawv kiag li cov qauv. Raws li ib tug txoj cai, txoj kev loj hlob ntawm hypnotic nyhuv tom qab thov tshuaj no yog tsim los rau 35-65 feeb thiab kav rau 6-9 teev.
Peb tsis tau hais tias cov tshuaj nyob rau hauv saib xyuas yuav teev cia cov lus hais rau anticonvulsant zog. Lawv tshwm sim los ntawm tus ntawm cov tshuaj nyob rau hauv tej qhov chaw ntawm lub paj hlwb. Thaum uas siv cov tshuaj no nyob rau hauv cov neeg mob tsis neuronal excitability nyob rau hauv epileptogenic tsam uas tsis pub cov emergence thiab kis ntawm pulses. Tsis tas li ntawd nyob rau hauv lub keeb kwm yav dhau ntawm "Luminal" hais tias thaiv cov hlab high-zaus ntswg ntawm neurons, lub nce nyob rau hauv lub chaw pib ntawm hluav taws xob stimulation nyob rau hauv lub cev muaj zog cheeb tsam ntawm lub cerebral cortex.
Nyob rau hauv tas li ntawd, rau qhov muab tshuaj yog yus muaj los ntawm ib tug me me analgesic nyhuv thiab antigiperbilirubinemichesky. Tsis tas li ntawd tsis kav tawm ntxiv dag zog rau ntawm lub cev txoj kev xav rau mob stimuli.
Me noj tshuaj npaum cas "luminal" muaj ib tug calming nyhuv, thiab siab -ugnetayut ua tsis taus pa medulla chaw zov me nyuam thiab t. D.
kev tig tau nta
seb cov tshuaj yog absorbed, "Luminal"? Cov lus qhia rau kev siv qhia tias hauv lub cev nws undergoes ib tug qeeb thiab ua kom tiav haum. Lub bioavailability ntawm tus neeg saib xyuas yog hais txog 80%, thiab cov ntawv cog lus rau ntshav cov nqaijrog - txog 30%.
Lub active ingredient ntawm cov tshuaj penetrates leej niam lub mis nyuj, raws li zoo raws li lub tsev me nyuam. Tsis tas li ntawd, nws muaj peev xwm muab faib nyob rau hauv lub me nyuam hauv plab ntaub so ntswg.
Feem "luminal" tshwm sim ntawm ob lub raum nyob rau hauv unchanged daim ntawv los yog nyob rau hauv daim ntawv ntawm cov metabolites. Rau phenobarbital yus heev cim cia hnab khib. Mob ntawm ob lub raum ua prolongation ntawm kev txiav txim.
Tshuaj "Luminal": indications rau kev siv
Xam tias yog ib tug yeeb tshuaj yog tshuaj tsis tau tsuas yog rau cov neeg laus, tab sis cov me nyuam thiab cov me nyuam mos. Raws li ib tug txoj cai, nws yog siv rau:
- hyperbilirubinemia;
- qaug dab peg;
- tetanus (rau adjuvant therapy);
- kev kho mob ntawm mob convulsive qaug dab peg.
Peb tsis tau hais tias qhov cuab tam yuav tau muab lub neej coj kev kho mob raws li ib tug sedative siv yeeb tshuaj nyob rau hauv thiaj li yuav tshem tawm cov kev ntxhov siab vim, kev ntshai thiab kev nyuaj siab.
Bans siv
Tam sim no koj paub nyob rau hauv dab tsi tej yam kev mob cov neeg mob cov kws kho ib yam tshuaj "Luminal". Indications rau kev siv ntawm cov tshuaj no tau teev tseg saum toj no. Nrog kev xav txog cov contraindications, ces lawv nqa xws li:
- siab rhiab heev mus rau yeeb tshuaj;
- mob loj heev siab thiab raum puas tsuaj;
- ntau yam ntaub ntawv ntawm porphyria;
- lactation thiab cev xeeb tub.
Medicament "Luminal": cov lus qhia rau kev siv rau cov me nyuam thiab cov laus
Kev siv cov tshuaj no yuav tsum tau nruj me ntsis qhia. Nws siv yuav tsum tau cov kev xaiv ntawm tus kheej kev kho mob regimen, ntau npaum, thiab ntev uas nyob tsis tau tsuas yog nyob rau hauv lub hom khiav ntawm tus kab mob, tab sis kuj nyob rau hauv tus neeg mob lub hnub nyoog thiab lwm yam ntxwv.
Raws li cov lus qhia, qhov nruab nrab ib koob tshuaj uas qhia cov cuab yeej rau cov neeg laus yog 10-200 mg. Noj xws tshuaj yuav tsum tau 1-3 zaug ib hnub twg.
Raws li rau cov me nyuam mos cov me nyuam, rau lawv cov tshuaj txhaj koob tshuaj yog muab xam rau ntawm lub cev qhov ceeb thawj (1-10 mg / kg lub cev hnyav ib hnub peb zaug).
Yog hais tias siv los kho cov kab mob hauv daim ntawv ntawm cov tshuaj Txoj kev lis ntshav, ntau npaum rau cov neeg laus yog 100-1400 mg (tso dej Txoj kev lis ntshav), los yog 10-200 mg (rau intramuscular txhaj).
Muab xam los ntawm koob tshuaj ntawm cov kev kawm ntawm cov me nyuam txoj kev noj tshuaj no kuj ua raws li nyob rau hauv tus me nyuam qhov kev hnyav.
Raws li cov kws txawj, tom qab tso dej thawj coj, "luminal" nws siab tshaj plaws cov nyhuv yog mus txog hauv 35 feeb.
phiv
Koj tsis zoo influences rau tib neeg lub cev tshuaj "Luminal"? Cov lus qhia rau kev siv (los ntawm ib tug kev tsis haum tshuaj nws txhais tau hais tias tsis qhia) cav hais tias cov kev kho mob ntawm cov ntaub ntawv ntawm cov tshuaj tus neeg mob tej zaum yuav tsim ib tug ntau yam ntawm cov kev phiv uas muaj feem xyuam tag nrho cov tseem ceeb heev nruab nrog cev thiab tshuab. Phiv cov tsos mob tsis muaj zog, qaug zog, tsaug zog, kev nyuaj siab thiab ataxia. Nws yog tseem tau txoj kev loj hlob ntawm thrombocytopenia, agranulocytosis, allergic kev tig cev thiab mob ntawm calcium metabolism.
tus neeg mob ntawm overdose
Nrog ib tug overdose ntawm "TMB" cov neeg mob heev feem ntau muaj mob taub hau, nystagmus, kiv taub hau, ataxia, ua tsis taus pa muaj teeb meem, nkees, tsis muaj zog, kev hais lus tsis zoo, koj nkees nkees, kev hloov nyob rau hauv lub cev kub, arousal, cov ntshav siab thiab lwm yam failures. Nyob rau hauv ntau txoj mob, muaj yog: bradycardia los yog tachycardia, pulmonary edema, tsis meej pem, arrhythmias, coma, mob ntsws thiab thiaj li nyob.
Yuav kom tshem tawm cov tsos mob no yog kws pais plab lavage li zoo raws li lub detoxification kev kho mob.
tshuaj cov kev sib tshuam
Daim ntawv thov ntawm qhov suav hais tias neeg sawv cev nyob rau hauv ua ke nrog tshuaj depressing HC, methylphenidate los yog Mao inhibitor tsub kom lub concentration ntawm nws active muaj nyob rau hauv nyob tus yeees ntawm cov ntshav, uas ua rau yus muaj zog tshuaj lom nyhuv thiab inhibition ntawm cov NA.
Lub ua ke ntawm "Luminal" nrog corticosteroids, chloramphenicol, corticotropin, dacarbazine, cyclosporine, digitalis glycosides, quinidine, metronidazole, tricyclic antidepressants, carbamazepine, anti-qaug dab peg, teej tug succinimides pab pawg neeg, doxycycline, anticoagulants, chlorpromazine, fenoprofenom, vitamin D thiab phenylbutazone yuav txo tau lub sij hawm kev txiav txim thiab kev siv ntawm cov tshuaj ua rau kom lawv metabolism, raws li zoo raws li lub nra rau lub siab.
Tib kev kho mob nrog acetazolamide yuav ua rau kom txoj kev loj hlob ntawm rickets thiab osteomalacia. Valproic acid tej phenobarbital concentration hauv cov ntshav, uas ua rau ib tug qhia tau tshuaj kom tsaug zog thiab nkees.
Siv "luminal" ua ke nrog nimodipine, "Verapamil" thiab felodipine thiaj li lawv concentration hauv cov ntshav.
Lub ua ke ntawm lub medicament nrog maprotiline tej nws inhibitory ntxim rau cov NA, thiaj li muaj cov nyhuv ntawm anticonvulsant barbiturates thiab convulsive chaw pib.
Active muaj "luminal" paracetamol tej zaum yuav txo efficiency thiab txhawb txoj kev loj hlob ntawm hepatotoxicity. Thaum ua ke nrog folic acid thiaj li efficiency ntawm phenobarbital.
Pyridoxine lowers ntshav concentration ntawm phenobarbital, thiab primidone, felbamate thiab, conversely, txhim khu nws.
Analogs ntawm cov tshuaj thiab nws cov nqi
Cov yooj yim tshuaj no yog analogues xws li "Barbinal" thiab "Dormiral".
Nqi ntsiav tshuaj "Luminal" (100 mg, 10 pcs.) Ntawm 1100 rubles thiab saum toj no.
tej ntaub ntawv
Tib mus txais tos "luminal" los ntawm ethanol thiab ethanol-txhais tau tias yuav ho txhim khu lub inhibitory nyhuv ntawm cov tshuaj nyob rau hauv lub paj hlwb ntawm tus neeg mob. Yog li ntawd, dej cawv thiab lwm yam lam tinctures rau haus dej haus cawv thaum lub sij hawm kev kho mob nrog rau cov ua hauj lawm yog txhob.
Xyuas
Feem ntau cov kev xyuas txog kev npaj no tawm rau cov niam txiv ntawm cov me nyuam yaus. Lawv cam tias cov tshuaj "Luminal" zoo sib ntaus nrog cov kab mob xws li qaug dabpeg thiab convulsive tej yam kev mob. Nws yog feem ntau kuj cov tshuaj no yog siv raws li ib feem ntawm kev ua ke nrog txoj kev kho, Nkij los txuam rau nws painkillers.
Muaj ntau cov neeg mob hais high efficiency ntawm cov tshuaj "Luminal". Txawm li cas los, lawv tam sim ntawd stipulated hais tias thaum tau txais daim ntawv ntawm cov nyiaj yuav tsum nruj me ntsis raws li cov tshuaj thiab nws ua ke nrog lwm yam tshuaj.
Tej zaum xam tau tias yog ib yam tshuaj uas siv rau cov kev kho mob ntawm cov neeg uas muaj vascular dystonia, uas yog nrog los ntawm bouts ntawm ntshai sib cem. Kev kho mob ntawm qhov cuab tam yuav pab tau normalize lub zwj ceeb ntawm cov neeg mob, tshwj xeeb tshaj yog yog hais tias nws yog ib tug ntxiv tshuaj, ceev cov hlab ntsha thiab relieves chua.
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