Noj qab haus huv, Npaj
Tshuaj "Mazeppa": cov lus qhia rau kev siv. Xyuas ntawm kev npaj "Medazepam"
Nyob rau hauv tej rooj plaub, cov tshuaj "Mazeppa" yuav siv tau? Nqe, indications thiab cov lus qhia ntawm cov tshuaj uas hais no hauv qab no.
Form, muaj pes tsawg leeg
"Mazeppa" - Ntsiav tshuaj puag ncig, Valium. Lawv yooj yim tshuaj yog Medazepam. Nrog kev xav txog ntxiv Cheebtsam, raws li lawv protrude starch, lactose monohydrate thiab calcium stearate.
nyhuv ntawm cov tshuaj
Yuav ua li cas yog cov tshuaj, "Mazeppa"? Cov lus qhia rau Siv hais tias nws yog ib qho anxiolytic neeg sawv cev, los yog lub thiaj li hu ua tranquilizer. Qhov no tshuaj yog ib tug derivative ntawm benzodiazepine. Nws exhibits anxiolytic, antiepileptic thiab nqaij relaxant yam ntxwv, thiab muaj ib tug bland timolepticheskoe nyhuv.
Hypnotic thiab sedative los ntawm cov tshuaj yog cai rau ib tus twg lesser tshaj nyob rau hauv cov pa benzodiazepine anxiolytics. Nyob rau hauv no hais txog, cov medicament nyob rau hauv lo lus nug hais txog ib tug txawv pab pawg neeg "nruab hnub" tranquilizers.
Qhov no tus neeg saib xyuas ua num ua ke nrog receptors (benzodiazepine) ntawm lub limbic system, raws li zoo raws li lub tsim ntawm ib tug activating uplink brainstem (lub hlwb). Ua tsaug rau nws, yog lub qhib ntawm chloride raws, uas thaum kawg ua rau yus muaj zog retarding nyhuv ntawm GABA nyob rau hauv lub Cns.
Tsis tas li ntawd nco ntsoov tias cov tshuaj "MAZEPA", cov lus qhia rau kev siv ntawm uas yog tau piav rau hauv qab no, yuav pab tau tshem tawm kev ntxhov siab vim, kev nyuaj siab psychoneurotic, ntxhov siab vim, nervousness thiab redundant general lub cev muaj zog stimulation. Nyob rau hauv tas li ntawd, nws yog ib lub stabilizing ntxim rau cov autonomic NS, restores kev xav coj tus cwj pwm thiab ib tug tseem ceeb soj ntsuam ntawm lawv tus kheej tus kab mob.
kinetics
Yuav ua li cas yog cov pharmacokinetic tsis yam ntxwv ntawm lub tranquilizer "Mazeppa"? Cov lus qhia rau Siv hais tias tom qab haus ntawm cov ntsiav tshuaj yog sai absorbed nyob rau hauv tus nqi ntawm cov 50-75%. Lawv siab tshaj plaws nyob rau hauv concentration cov ntshav mus txog ob teev tom qab. Ruaj rau ntshav ntshav protein yog 99,7%.
Metabolites yog muab tau los ntawm txhais tau tias ntawm ob lub raum thiab nyob rau hauv cov hnyuv rau 20-175 teev.
zaj lus tim khawv
Ntsiav tshuaj "Mazeppa", xyuas uas koj yuav nrhiav tau hauv qab no, siv rau irritability, nervousness, pog thiab tshee nro. Nws kuj pom zoo kom siv cov txhais tau tias nyob ntsoos ntsoos cov tsos mob rau cov neeg uas raug kev txom nyem los ntawm alcoholism, los mus tiv thaiv yastes yastaw thiab lawm syndrome.
Nyob rau hauv paediatrics tshuaj no yog siv kom muaj zog excitability ntawm tus me nyuam, puas siab puas ntsws lability thiab "lub tsev kawm ntawv" neuroses.
Contraindications
Cov kev kawm txhais tau tias yuav tsum tsis txhob noj thaum uas cev xeeb tub, myasthenia Heavy kev, "Hmo ntuj" apnea medazepama intolerance, pathologies ntawm lub raum thiab lub siab, pub niam mis thiab ntau yam ntaub ntawv nyob (tshuaj, haus dej cawv). Tsis tas li ntawd, active tshuaj yog ua rau cerebellar ataxia, organic pathology HC, ocular tawg, ua pa tsis ua hauj lwm thiab tus txha caj ataxia.
Tranquilizer "Mazeppa": cov lus qhia rau kev siv
"Medazepam" Ntsiav tshuaj yog npaum li cas peb lub sij hawm ib hnub twg, pib nrog ib tug tsawg koob tshuaj yog 5 mg. Maj mam tus nqi ntawm cov tus neeg saib xyuas yog tom mus rau 30 mg ib hnub twg. Nyob rau hauv tsawg tus neeg mob, pub rau noj 40 mg ntawm cov tshuaj ib hnub twg.
Nyob rau hauv mob kev kho mob yog pom zoo hais tias cov nram qab no kev kho mob tswvyim: 5 mg ntawm yeeb tshuaj nyob rau hauv lub yav sawv ntxov thiab 10 mg - yav tsaus ntuj. Nyob rau hauv lub tsev kho mob txhua hnub nyiaj pab ntau tshaj ntau npaum ntawm no neeg sawv cev yuav tau nce mus 60-70 mg.
Lub caij ntawm qhov kev kho no neeg sawv cev yog 2 lub hlis (nyiaj pab ntau tshaj). Tom qab 30 hnub, cov kev yuav tau rov qab.
phenomena sab
Cov kev kawm yuav ua rau cov hauv qab no los:
- dyspepsia, nce bilirubin, AST, ALT, qhov ncauj qhuav;
- tachycardia, ntshav siab poob;
- stupor, disinhibition, mob taub hau, anterograde amnesia, kev pab paresis, kev nyuaj siab, kiv taub hau, dysarthria, qaug zog, tsis meej pem, ataxia, aggression, tsis meej pem;
- nyob rau hauv cov neeg uas muaj COPD thaum noj siab koob tshuaj ntawm cov tshuaj cai alveolar hypoventilation;
- rhuav txhua ntawm cov pa ib ntsuj av tau thiab lub hlwb puas tsuaj cai inhibition ntawm cov pa chaw.
tej tswv yim pom zoo
Ntsiav tshuaj "Medazepam" tej zaum yuav ua rau kom muaj kev cuam tshuam ntawm cov xim thiab nco, raws li zoo raws li lub yuav txo tau txoj kev kawm.
Ua ke nrog rau kev siv impermissible txhais tau tias etanolsoderzhashih dej qab zib.
Nws pom zoo kom ib tug gradual tshem ntawm cov tshuaj nyob rau hauv cov kev kho mob ntawm ntsoos ntsoos cov tsos mob.
Heev txoj kev kho yuav tsim tshuaj quav medozepama.
Nqe thiab kev txheeb xyuas
Nqi saib xyuas tranquilizer yog hais txog 150 rubles.
Testimonials qhia zoo zoo nkauj tolerability ntawm cov tshuaj nyob rau hauv raws li nrog tag nrho cov lus qhia ntawm tus kws kho mob thiab cov dosing regimen. Txawm tias nyob rau hauv ib tug ob peb tus neeg mob no txhais tau tias tsis tau yeej txhawb tshuaj tiv, yuav txo tau ntawm potency, urinary tuav, paradoxical tshua, kev tsis haum tshuaj, mob hauv siab thiab dysmenorrhea.
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