Noj qab haus huvNpaj

"Flyuanksol": cov lus qhia rau kev siv, tiag tiag cov kws kho mob. Sab los "Flyuanksola" analogues ntawm cov tshuaj

Yuav ua li cas yog cov tshuaj "Flyuanksol"? Cov lus qhia rau kev siv ntawm cov tshuaj, nws cov khoom xyaw, phiv, qhov kev tso tawm daim ntawv thiab pharmacological khoom no piav nyob rau hauv kom meej nyob rau hauv no tsab xov xwm. Los ntawm nws koj yuav kawm txog dab tsi lub contraindications thiab indications tau hais tias cov tshuaj, ntau npaum li cas nws cov nqi, yuav ua li cas nyob rau hauv cov ntaub ntawv ntawm ib tug overdose, thiab hais txog. D.

Muaj pes tsawg leeg ntawm cov tshuaj thiab nws tso tawm ntaub ntawv

Yuav ua li cas yog lub active tshuaj muaj cov tshuaj "Flyuanksol"? qhia rau kev siv ntawm lub medicament phau ntawv hais tias raws li active tivthaiv nws protrudes flupenthixol hydrochloride.

Raws li rau hauv daim ntawv ntawm kev tso tawm, tab sis hnub no nws yog ib tug txhais tau tias yuav tsum pom xwb nyob rau hauv dauv, ntsiav tshuaj thiab cov tshuaj, ib tug roj-raws li, npaj rau intramuscular thawj coj. Tus thawj tshuaj no yog marketed nyob rau hauv lub khob zatemennom 10 ml, ib tug thib ob - nyob rau hauv ib tug thawv 100 los yog 50 thiab peb - nyob rau hauv ampoules ntawm 10 daim.

General thaj chaw ntawm cov tshuaj

Yog vim li cas yog tshuaj "Flyuanksol"? Testimonials txog cov tshuaj no yog hais hauv qab no. Ntsiav tshuaj thiab txhaj tshuaj yog ib pab pawg neeg ntawm antipsychotics. Lawv muaj anxiolytic, antidepressant thiab sedative nyhuv. Zoo tswv yim txog cov tshuaj no muaj cov ntaub ntawv uas nws nraaj activates lub siab ntsws lub xeev ntawm tus neeg mob thiab txhawb rau kev adaptation.

Lub pharmacological cov yam ntxwv ntawm cov tshuaj

Yuav ua li cas yog cov yam ntxwv ntawm pharmacological tshuaj "Flyuanksol"? Cov lus qhia rau kev siv qhia tias cov tshuaj no yog ib tug neuroleptic, thaiv cov hlab adrenergic receptors thiab dopamine receptors nyob rau hauv lub hlwb. Raws li ib tug tshwm sim ntawm lub active tshuaj yog tiav tshuaj kom tsaug zog. Feem ntau, qhov no tshwm sim tshaj ib tug 8-hnub kev npaum li cas.

Yuav ua li cas cov neeg mob txog cov tshuaj "Flyuanksol"? Xyuas ntawm cov neeg mob muaj ntau ntawm nthuav cov ntaub ntawv. Nyob rau hauv feem ntau tus neeg mob, lawv nco ntsoov hais tias cov tshuaj es sai sai eliminates tej yam tshwm sim ntawm psychosis thiab kev nyuaj siab, raws li tau zoo raws li yuav pab tau tus restoration kev xav. Cov neeg mob uas tau antisocial mob, yog sociable thiab hloov mus rau lub koom txoos.

nta tshuaj

Yuav ua li cas puas cov tshuaj "Flyuanksol"? Xyuas cov kws kho mob thiab lwm yam tshwj xeeb hais tias ib tug feature ntawm cov khoom no yog lus dag nyob rau hauv lub fact tias, nyob ntawm seb cov tshuaj nws tau ua nyob rau hauv tus neeg mob txawv.

Antipsychotic nyhuv manifests tom qab medicament daim ntawv thov txhais tau tias nyob rau hauv ib tug npaum li ntawm 3 mg ib hnub twg. Los ntawm txoj kev, cov kev siv ntawm tej yam tsub kom nrog lub noj tshuaj npaum cas.

Raws li uas mus txog rau 25 mg ib hnub twg cov tshuaj tsis muaj sedative nyhuv. Txawm li cas los, nws yuav tsum tau muab sau tseg tias nyob rau hauv ntau dua koob tshuaj, nws yuav ua uas tsis yog-kev sedative los.

Nyob rau hauv lub koob ntau yam xws neuroleptic neeg sawv cev muaj ib tug qhia tau anxiolytic nyhuv. Thaum uas siv cov me me koob tshuaj (nce txog li 3 mg ib hnub twg), cov tshuaj yuav pab raws li ib tug pa antidepressant tshuaj.

Yog li, cov tshuaj "Flyuanksol" yog tau txo lub ntsiab ntawm cov tsos mob psychosis, xws li paranoid delusions, hallucinations thiab xav tsis meej. Nws muaj disinhibitory zog (i.e. activating thiab antiautisticheskim) thiab thiaj li ib tug mus ob peb vas teeb meem, uas thaum kawg yeej txhawb kom cov neeg mob uas muaj depressive cov tsos mob, lawv cov kev sib adaptation tswj thiab tej sociability.

Ntxiv txog injectable daim ntawv

Kev npaj "Flyuanksol Depot" yog ib cov roj tov npaj rau intramuscular depot tshuaj. Nyob rau hauv lwm yam lus, cov tshuaj no yog tso daim ntawv flupenthixol.

Thaum uas siv cov tshuaj no nyob rau hauv me me thiab medium koob tshuaj (txog li 100 mg txhua txhua 14 hnub) rau tus neeg mob yog tsis unspecific tshuaj kom tsaug zog. Txawm hais tias nws yog tseem loj hlob nyob rau high school koob tshuaj.

Yuav ua li cas cov kws txawj hais txog daim ntawv no ntawm cov tshuaj ( "Flyuanksol Depot")? Xyuas muab hais tias xws li ib tug tov muaj ib tug ntev ntev raug rau tus neeg mob, es tsis tshuaj ntsiav tshuaj. Ntxiv mus, ua tsaug rau nws, nws yog ib qho yooj yim mus nqa tawm tas mus li antipsychotic kev kho mob, uas yog tsis tshua muaj ib qho tseem ceeb rau cov neeg mob uas tsis nqa tawm kev kho mob tshuaj.

Los ntawm cov saum toj no nws yuav xaus lus tias cov tshuaj "Flyuanksol Depot" yog tau los mus tiv thaiv heev rov txuam nrog txawj kev cuam tshuam ntawm txoj kev kho. Intramuscular txhaj yuav nqa tawm ntawm ua mib ntawm ob los yog plaub lub lis piam.

tshuaj

Yuav ua li cas tau ntev absorbed tshuaj "Flyuanksol"? Tom qab qhov ncauj thawj coj lub siab tshaj plaws concentration ntawm lub active caij yog tiav nyob rau hauv txog 3-7 teev nyob rau hauv ntshav. Lub bioavailability ntawm cov tshuaj yog 40%.

Active tshuaj caij me ntsis penetrates rau hauv lub placental barrier. Nws yuav tsum tau muab sau tseg tias, nyob rau hauv me me, nws yog tseem ceeb nrog niam cov kua mis. Incidentally, lub metabolites muaj neuroleptic kev ua si.

Yuav ua li cas puas txhaj "Flyuanksol Depot"? Phau Ntawv Qhia hais tias tom qab intramuscular txhaj ntawm yeeb tshuaj cis (Z) -flupentixol decanoate undergoes cleavage (enzymatic). Qhov no ntaub ntawv lub active caij ntawm lub cis (Z) -flupentixol thiab decanoic acid. Qhov siab tshaj plaws nyob rau hauv concentration ntshiab tau thawj los ntawm tus kawg ntawm lub thawj lub lim tiam tom qab txhaj tshuaj.

Thaum tau txais cov ntsiav tshuaj mus rau hauv lawv cov chaw ua taus zes lub sij hawm yog hais txog 35 teev. Yog hais tias muaj tau siv ib tug tov rau txhaj, lub concentration txo exponentially nyob rau hauv lub ntshiab (tom qab 3 lub lim tiam).

Tso tawm active medicament nyob rau hauv daim ntawv ntawm cov metabolites los ntawm cov hnyuv, thiab ob lub raum.

Indications rau kev siv ntawm neuroleptic cov neeg ua hauj

Nyob rau hauv tej rooj plaub, cov tshuaj qhia tau hais tias "Flyuanksol"? Nws txiav txim tej zaum yuav sib txawv, nyob ntawm seb ntau npaum.

Cov tshuaj no yog qhia nyob rau ntawm lub koob mus rau 3 mg ib hnub twg rau cov nram qab no pathological tej yam kev mob:

  • kev nyuaj siab me me thiab loj tsawv degree, nrog qaug zog, ntxhov siab vim thiab tsis muaj kev teg num;
  • psychosomatic mob uas tshwm sim nrog asthenic tshua;
  • neurotic mob (mob), nrog los ntawm apathy, kev nyuaj siab thiab ntxhov siab vim;
  • thiab mob situational ntxhov siab vim kev ntshawv siab, raws li tau zoo raws li lub xeev ntawm ntau kev ntxhov siab, tsis txhob yuav tsum tau ib tug sedative los yog hypnotic nyhuv (piv txwv li, yog hais tias tus neeg mob yog txhob tranquilizers).

Medicament "Flyuanksol", analogues ntawm uas yuav tsum tau nthuav tawm nyob rau thaum xaus ntawm qhov tsab xov xwm, yog tsa nyob rau ntawm lub noj tshuaj npaum cas ntawm 3 mg ib hnub twg thiab ntau hais tias muaj yog ib tug txawv ntawm cov hauv qab no: psychotic tej yam kev mob uas nrog paranoid delusions, hallucinations, teeb nyob rau hauv kev xav, anergy, apathy thiab tsi txawj has lug.

Contraindications rau kev siv ntawm neuroleptic cov neeg ua hauj

Nyob rau hauv tej rooj plaub, nws yog tsis pom zoo kom siv cov tshuaj "Flyuanksol"? Cov lus qhia rau kev siv muaj xws li cov nram qab no daim ntawv teev cov contraindications:

  • cov me nyuam lub hnub nyoog (18 xyoo);
  • Cns kev nyuaj siab;
  • lactation;
  • thaum lub sij hawm cev xeeb tub;
  • intoxication (mob) barbiturates;
  • cev qhuav dej;
  • intoxication mob opioid analgesics;
  • pheochromocytoma;
  • alcoholic mob lom;
  • raw lub xeev;
  • hloov hlwb pob txha hluav;
  • pathological kev hloov nyob rau hauv cov ntshav;
  • npau taws me ntsis rau neuroleptics muaj tioksantenoviy qauv.

Nws yuav tsum tau muab sau tseg tias cov tshuaj yog tsis pom zoo rau siv nyob rau hauv me me noj tshuaj npaum cas (3 mg) nyob rau hauv ib lub xeev ntawm hyperactivity los yog excitations.

Tshuaj "Flyuanksol": kev qhia (cov ntsiav tshuaj, dauv)

Rau cov kev kho mob ntawm kev ntxhov siab vim thiab kev nyuaj siab mob thawj zaug koob ntawm cov medicament nyob rau hauv lub ntsiav tshuaj yuav tsum yog 1 mg ib zaug ib hnub twg (nyiam dua nyob rau hauv lub yav sawv ntxov), los yog 500 mcg ib hnub ob zaug. Yog hais tias lub kho nyhuv yog tsis tuaj kawm ntawv, tus nqi ntawm cov tshuaj nyob rau hauv ib lub lim tiam yuav muab ntau zog rau 2 mg. Yog li lub hnub ntau npaum (2-3 mg) tau muab faib mus rau hauv ob peb ua sawv. Yog hais tias cov nyhuv yog tsis tuaj kawm ntawv thaum uas siv cov tshuaj nyob rau hauv lub maximal koob tshuaj (i.e., 3 mg), ces nws yuav tsum tau poob mus li.

Nyob rau hauv cov kev kho mob ntawm psychotic tej yam kev mob teem nqi ntawm cov tshuaj tsuas ib lub zuj zus. Thawj zaug txhua txhua hnub ntau npaum yuav tsum 3-15 mg nyob rau hauv 3 faib koob tshuaj. Yog hais tias qhov kev kawm, tus hais tias volume yuav muab ntau zog mus rau 20 los yog 30 mg ib hnub twg. Qhov siab tshaj plaws ntau npaum yuav tsum tsis txhob yuav ntau dua 40 mg.

Raws li sawv cev txij nkawm kho mob tus neeg saib xyuas yog muab nyob rau hauv ib tug npaum li ntawm 5-20 mg ib hnub ib zaug (nyob rau hauv lub yav sawv ntxov).

Raws li rau txoj kev nco "Flyuanksol", lawv yuav tsum tsuas yog noj hauv tsev. Cov kws kho mob feem ntau yog muab cov tshuaj nyob rau hauv daim ntawv no yog nyob rau hauv rooj plaub yog hais tias, txawm yog vim li cas, tsis tau noj cov tshuaj hais ntawm ncauj (ntsiav tshuaj). Supportive ntau npaum rau cov neeg mob yog 4-40 mg ib hnub twg.

Txhaj "Flyuanksol": kev qhia, ua siab ntev xyuas

Cov oily tov rau intramuscular depot tshuaj yuav tsum tau muab sib sib zog nqus mus rau hauv lub qaum txheej quadrant ntawm lub pob tw. Ntau npaum thiab lub luv ntawm kev kho mob yuav tsum tsuas yog ntsia ib lub zuj zus (ywj siab ntawm kho nyhuv).

Qhov no formulation yog feem ntau yog siv nyob rau hauv ib tug npaum li ntawm 20-40 mg (los yog 1-2 ml) txhua txhua 2 los yog 4 lub lis piam. Nws yuav tsum tau muab sau tseg tias ib txhia cov neeg mob yuav tsum tau loj koob tshuaj thiab lub luv luv luv ntawm tshuaj.

Yog hais tias cov hoob ntim cov tshuaj rau kev txhaj tshuaj (20 mg / ml) yog xav paub ntau tshaj 2 los yog 3 ml rau 1 txoj kev, nws yog tsim nyog los mus rau nrog cov tshuaj ntawm siab concentration.

Kev npaj ntawm 100 mg / ml yuav tsum tau txhaj nyob rau hauv ib tug ntim ntawm 50-200 mg (los yog 0.5-2 ml) txhua txhua 2-4 lub lis piam. Nyob rau hauv mob relapse los yog exacerbation ntawm tus kab mob tej zaum yuav tsum tau ib tug ib tug-lub sij hawm cov kev taw qhia nyob rau hauv txhais tau tias ib tug npaum li txog li 400 mg ntawm ua mib ntawm 2 los sis 1 lub lim tiam. Tom qab lub mob cov tsos mob dhau, koj yuav tsum tsim ib gradual yuav txo tau nyob rau hauv ntau npaum mus rau ib tug txij nkawm (20-200 mg txhua txhua 2-4 lub lis piam).

Yog hais tias yuav tsum tau mus dhau los ntawm lub qhov ncauj hauv daim ntawv ntawm cov tshuaj rau parenteral npaj txhawb txoj kev kho, nws yog pom zoo kom yuav tsum tau raws li nyob rau hauv cov nram no tswvyim:

  • txhua txhua hnub ntau npaum li cas (nyob rau hauv mg) ntawm cov tshuaj nyob rau hauv lub ntsiav tshuaj x 4 = ib ntau npaum (nyob rau hauv mg) txhaj tshuaj txhua txhua 14 hnub.

Nws yuav tsum tau muab sau tseg tias tsis pub dhau ib lub lim tiam tom qab thawj coj ntawm cov tshuaj yuav tsum tau mus ntxiv noj cov tshuaj nyob rau hauv cov ntsiav tshuaj, tab sis nyob rau hauv ib tug qis koob tshuaj. Ua raws li-up ntim thiab cov kis ntawm tus txheej txheem tsim nyob rau hauv raws li kho nyhuv.

Maximum ntau npaum injectable tshuaj (ib-theem) yog hais txog 400 mg. Yog li cov kis ntawm cov tshuaj yuav tsum yog nyob rau ntawm ib lub lim tiam.

Raws li cov lus teb ntawm cov neeg mob, thaum uas siv kom zoo, cov kev npaj thiab ua kevcai nco txog kev kho mob cov tswv yim, nws muaj ib tug zoo ntxim rau lawv tag nrho lub siab lub ntsws lub xeev.

phiv

Tau ib tug tsis zoo ntxim rau lub cev cov tshuaj "Flyuanksol"? Sab los yog tam sim no nyob rau hauv cov tshuaj, tsis hais txog ntawm nws daim ntawv. Ntawm no lawv yog tam sim no.

  1. Lub paj hlwb: giperkinetiko-hypertensive syndrome (extrapyramidal teeb), tsis muaj zog, akathisia, nkees, kiv taub hau, psychomotor ruamqauj, tardive dyskinesia, dystonic tshua thiab neuroleptic phem syndrome.
  2. Lub plawv thiab cov hlab ntsha: tachycardia, hypotension, orthostatic.
  3. hematopoietic system: granulocytopenia.
  4. Kev txiav txim zoo hauv nruab nrog cev: disturbance ntawm kev pab.
  5. GI: cem quav, jaundice cholestatic, qhov ncauj qhuav, nraum hloov nyob rau hauv daim siab muaj nuj nqi kev ntsuam xyuas.
  6. Endocrine system: qhov hnyav nce, galactorrhea, tawm hws, gynaecomastia, impotence, dysmenorrhea, nce qab los noj mov, poob libido, kub flashes.
  7. Mob txeeb system: urinary tuav tseg.
  8. Kev ua xua: dermatitis, photosensitivity, thiab daim tawv nqaij pob.

Tshwj xeeb cov lus qhia rau kev siv

Nrog huab ceev faj tshuaj rau cov neeg mob nrog plawv mob, convulsive mob, ua pa tsis ua hauj lwm, glaucoma, Parkinson tus kab mob, mob plab ulcers thiab 12-tiperstnoj hnyuv, mob hawb pob, alcoholism, mob hawb pob, mob txeeb tuav, daim siab tsis ua hauj lwm, thiab benign prostatic hyperplasia.

Yog hais tias tus neeg mob tau yav tas los tau txais neuroleptics los yog tranquillizers nrog sedative nyhuv, nws yog tsim nyog los tsis txhob noj lawv ntseeg nkaws.

Thaum ntev-lub sij hawm kev kho mob, tshwj xeeb tshaj yog nyob rau high school noj tshuaj npaum cas pom zoo los tswj thiab ntsuam xyuas tus neeg mob tus mob nyob rau hauv thiaj li yuav kho txij nkawm koob tshuaj.

Nyob rau hauv lub simultaneous kev kho mob ntawm cov ntshav qab zib hauj lwm ntawm hais tias formulation yuav tsum tau kho tus nqi ntawm cov kua dej los.

Nyob rau hauv daim ntawv thov ntawm neuroleptics yuav tsim neuroleptic phem syndrome. Nws lub ntsiab tsos mob nqaij rigidity, hyperthermia, kho kev puas hlwb raws li txoj cai, thiab ua hauj lwm ntawm lub autonomic lub paj hlwb. Thaum xws li cov tsos mob yuav tsum tau ceev tshem tawm ntawm lub sij hawm ntawm cov tshuaj thiab txhawb symptomatic kev kho mob.

Nyob rau hauv feem ntau tus neeg mob, cov tshuaj "Flyuanksol" tsis ua kom loog. Tab sis, dua li no, nws yog tsim nyog los noj mus rau hauv tus account nws tej yam nyob rau hauv lub peev xwm los xyuam xim khiav lag luam hauv lub tshuab, los yog lwm yam mechanisms. Kuv kuj xav kom nco ntsoov tias thaum lub sij hawm txoj kev kho (tshwj xeeb tshaj yog nyob rau hauv lub pib), cov neeg mob yuav tsum tsis txhob muaj feem tej chaw ua hauj lwm (los txiav txim seb cov lus teb mus rau yeeb tshuaj).

tus neeg mob ntawm overdose

Yog hais tias cov tshuaj yog coj kom zoo (nce volume), tej zaum nws yuav tshwm sim overdose. Nyob rau hauv cov ntaub ntawv no, exhibits lub nram qab no cov yam ntxwv: hypo- los yog hyperthermia, nkees nkees, convulsions, extrapyramidal teeb meem, kev poob siab, hypotension thiab coma.

Yuav ua li cas nyob rau hauv xws li ib tug teeb meem no? Nws yog tsim nyog los nqa tawm ib tug txhawb thiab symptomatic txoj kev kho. Yog hais tias cov tshuaj tau noj, yuav tsum tau mus sai sai ntxuav tawm lub plab, raws li zoo raws li yuav lub sorbent. Nyob rau hauv tas li ntawd, nws tseem ceeb heev los pab txhawb cov kev ua ub ntawm cov hlab ntsha, lub plawv thiab ua pa system. Nws tsis pom zoo kom siv epinephrine raws li nws tej zaum yuav ua rau cov ntshav siab yuav txo tau. Extrapyramidal cov tsos mob yog tau kom txhob muaj cov tshuaj "Biperiden" thiab qaug dab peg - "Diazepam".

Sis nrog lwm yam tshuaj

Thaum siv ib tug theem ntawm hais tias medicament tej zaum yuav amplified sedative los ntawm barbiturates, ethanol, thiab lwm yam tshuaj mas siv uas muaj inhibitory ntxim rau cov Cns.

Kev npaj "Flyuanksol" nws yog tsis pom zoo siv nyob rau hauv ua ke nrog guanethidine thiab Drug tshuaj nrog ib tug zoo xws li cov nyhuv. Qhov tseeb yog vim lub fact tias antipsychotics tej zaum yuav heev tsis muaj zog txaus lawv antihypertensive los.

Nrog ib leeg-siv medicament "Flyuanksol" nws yuav txo tau miv nyuas siv zug ntawm cov tshuaj "levodopa" thiab lwm yam adrenergic agents.

Nyob rau tib lub sij hawm noj cov tshuaj nrog ib tug "piperazine" thiab "MCP" ho tsub kom kev pheej hmoo ntawm extrapyramidal teeb meem.

Nws yuav tsum tau muab sau tseg tias neuroleptic tshuaj hais raws li ib tug tshuaj cov kev txhaj tshuaj nyob rau hauv txhua rooj plaub yuav tsum tsis txhob yuav tov nrog rau lwm cov kua.

Nqe thiab analogues ntawm cov tshuaj

Yuav ua li cas npaum li cas yog ib tug yeeb tshuaj "Flyuanksol"? Nws nqi yog heev siab heev. Yog li ntawd, rau 50 ntsiav tshuaj ntawm 1 mg ntawm koj yuav tau them txog 500 Lavxias teb sab rubles. Yog hais tias koj xav tau 100 5 mg cov ntsiav tshuaj, lawv yuav tsum tau muas 1,200 rubles. Raws li rau lub tshuaj daim ntawv ntawm cov tshuaj, nws yog txawm ntau kim heev. Tshaj 10 vials (20 mg / ml) pharmacists yuav tsum tau hais txog 2300 rubles.

Yuav ua li cas yog hais tias tus neeg mob yog tsis mus yuav tshuaj "Flyuanksol"? Nws analogues yog muag nyob rau hauv yuav luag tag nrho cov khw muag tshuaj chains. Ntawm lawv yog cov hauv qab no:

  1. Cov tshuaj "Flyuanksol Depot". Qhov no yog ib tug ceev thiab ntau haib siv yeeb tshuaj. Txawm li cas los, nws yog ntau npaum li cas kim ntsiav tshuaj.
  2. "Klopiksol" tshuaj. Nyob rau hauv tus nqi yog heev ze rau tus thawj. Nws mus rau khoom nyob rau hauv lub ntsiav tshuaj thiab muaj ib tug ob peb contraindications.
  3. "Truksal" txhais tau tias. Muag nyob rau hauv cov ntsiav tshuaj. Lub ntsiab kom zoo dua nyob rau hauv dej siab ntawm txoj kev siv rau cov me nyuam nrog 3-xyoos. Nqi me ntsis saum toj no tseem cia nrog.

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